SCHEMBL8538985

SCHEMBL8538985

O=S(=O)(c1ccccc1)c1ccc(Nc2ncnc3cc(CCCCN4CC[S+]([O-])CC4)ccc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.47
AURKA O14965 9/20 0.46
AURKB Q96GD4 9/20 0.46
SUV39H1 O43463 2/20 0.43
ERBB2 P04626 1/20 0.41
KDR P35968 2/20 0.40
PRMT1 Q99873 1/20 0.40
SMYD3 Q9H7B4 1/20 0.40
HSD17B10 Q99714 1/20 0.39
BRAF P15056 1/20 0.39
TNNI3K Q59H18 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8367738 0.97 EGFR (0.47) EGFRAURKAAURKBSUV39H1ERBB2
SCHEMBL8541789 0.93 EGFR (0.47) EGFRAURKAAURKBERBB2KDR
SCHEMBL8363554 0.91 EGFR (0.47) EGFRAURKAAURKBERBB2KDR
SCHEMBL8516124 0.87 EGFR (0.49) EGFRAURKAAURKBSUV39H1ERBB2
SCHEMBL8545642 0.86 EGFR (0.47) EGFRAURKAAURKBERBB2KDR
SCHEMBL8365522 0.84 EGFR (0.47) EGFRAURKAAURKBERBB2KDR
SCHEMBL8364953 0.84 AURKA (0.55) EGFRAURKAAURKBERBB2KDR
SCHEMBL8367261 0.83 EGFR (0.55) EGFRAURKAAURKBERBB2
SCHEMBL8367320 0.83 EGFR (0.54) EGFRAURKAAURKBERBB2KDR
SCHEMBL8364112 0.82 EGFR (0.62) EGFRAURKAAURKBERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999035132-A1 HETEROCYCLIC COMPOUNDS GLAXO GROUP LIMITED (GB) 1999-07-15 WO disclosed