SCHEMBL8539210

SCHEMBL8539210

C[C@@H](n1ccn(-c2ccc(OC(F)(F)C(F)F)cc2)c1=O)[C@](O)(Cn1cncn1)c1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 11/20 0.42
CYP2C9 P11712 11/20 0.42
CYP2C19 P33261 11/20 0.42
CYP1A2 P05177 5/20 0.42
CYP2D6 P10635 5/20 0.42
KCNH2 Q12809 1/20 0.42
KMT2A Q03164 1/20 0.39
LMNA P02545 2/20 0.38
CYP2B6 P20813 1/20 0.38
CYP3A5 P20815 1/20 0.38
CYP3A7 P24462 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP3A43 Q9HB55 1/20 0.38
CYP46A1 Q9Y6A2 1/20 0.38
MAPT P10636 1/20 0.34
HSP90AA1 P07900 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
ADRA1A P35348 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8538916 0.91 CYP3A4 (0.40) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8097544 0.89 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9231939 0.87 CYP3A4 (0.40) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9232008 0.87 CYP3A4 (0.41) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8106906 0.87 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8105389 0.87 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9229215 0.82 CYP2C19 (0.39) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8540421 0.82 CYP3A4 (0.57) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8539997 0.82 KMT2A (0.39) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8535041 0.81 CYP3A4 (0.59) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792780-A FUNGICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-08-11 US disclosed
EP-0657449-B1 Azole compounds, their production and use as antifungal agents TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-04-08 EP disclosed
US-5545652-A Triazole and imidazole compounds and their use as antifungal therapeutic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-08-13 US disclosed
EP-0657449-A1 Azole compounds, their production and use as antifungal agents Takeda Chemical Industries, Ltd. (JP) 1995-06-14 EP disclosed