SCHEMBL9232008

SCHEMBL9232008

C[C@@H](n1cnn(-c2ccc(OC(F)(F)C(F)F)cc2)c1=O)[C@](O)(Cn1cncn1)c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 13/20 0.41
CYP2C9 P11712 12/20 0.41
CYP2C19 P33261 12/20 0.41
CYP1A2 P05177 6/20 0.41
CYP2D6 P10635 6/20 0.41
KCNH2 Q12809 3/20 0.41
KMT2A Q03164 1/20 0.40
LMNA P02545 2/20 0.37
CYP2B6 P20813 1/20 0.37
CYP3A5 P20815 1/20 0.37
CYP3A7 P24462 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP3A43 Q9HB55 1/20 0.37
CYP46A1 Q9Y6A2 1/20 0.37
HSP90AA1 P07900 2/20 0.34
CYP19A1 P11511 2/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
ADRA1A P35348 1/20 0.34
CYP51A1 Q16850 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9229186 0.90 CYP3A4 (0.40) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8105672 0.89 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8539210 0.87 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9226049 0.87 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9231939 0.85 CYP3A4 (0.40) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9229215 0.83 CYP2C19 (0.39) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8539997 0.82 KMT2A (0.39) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8718366 0.82 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8718513 0.80 CYP3A4 (0.61) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8718383 0.80 CYP3A4 (0.57) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0659751-A1 Optically active azole derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-06-28 EP disclosed