SCHEMBL8540466

SCHEMBL8540466

COCC1(COC)Oc2ccc(C#N)cc2[C@@H](Nc2ccc(=O)n(CC3CC3)n2)[C@@H]1O

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 8/20 0.40
ABCB1 P08183 10/20 0.38
ABCC8 Q09428 2/20 0.35
KCNJ11 Q14654 2/20 0.35
KCNJ8 Q15842 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8537349 0.91 ABCC9 (0.41) ABCC9ABCB1
SCHEMBL8535817 0.90 ABCC9 (0.41) ABCC9ABCB1
SCHEMBL8536345 0.89 ABCC9 (0.40) ABCC9ABCB1CYP1A2CYP2D6CYP2C19
SCHEMBL8535230 0.89 ABCC9 (0.42) ABCC9ABCB1
SCHEMBL8538266 0.89 ABCC9 (0.40) ABCC9ABCB1
SCHEMBL8537101 0.89 ABCB1 (0.41) ABCC9ABCB1
SCHEMBL8539533 0.89 ABCC9 (0.40) ABCC9ABCB1
SCHEMBL8535712 0.89 ABCC9 (0.41) ABCC9ABCB1
SCHEMBL8540184 0.88 ABCC9 (0.39) ABCC9ABCB1CYP1A2CYP2D6CYP2C19
SCHEMBL8539755 0.88 ABCC9 (0.39) ABCC9ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719155-A CARDIOVASCULAR DISORDERS JAPAN TOBACCO INC. (JP) 1998-02-17 US claimed
EP-0677519-A1 CHROMAN DERIVATIVE AND MEDICINAL USE THEREOF Japan Tobacco Inc. (JP) 1995-10-18 EP claimed
US-5719155-A CARDIOVASCULAR DISORDERS JAPAN TOBACCO INC. (JP) 1998-02-17 US disclosed
EP-0677519-A1 CHROMAN DERIVATIVE AND MEDICINAL USE THEREOF Japan Tobacco Inc. (JP) 1995-10-18 EP disclosed