SCHEMBL8540506

SCHEMBL8540506

CC(C)[C@H](NC(=O)NCc1ccccc1)C(=O)NC(Cc1ccccc1)C(O)C(Cc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 10/20 0.58
CTSD P07339 2/20 0.57
KLK5 Q9Y337 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7269992 0.89 CTSD (0.61) BACE1CTSD
SCHEMBL8532173 0.87 KLK5 (0.61) BACE1CTSDKLK5
SCHEMBL8531207 0.87 KLK5 (0.61) BACE1CTSDKLK5
SCHEMBL6447745 0.85 CTSD (0.66) BACE1CTSDKLK5
SCHEMBL7268902 0.84 KLK5 (0.61) BACE1CTSDKLK5
SCHEMBL7270278 0.84 CTSD (0.67) BACE1CTSDKLK5
SCHEMBL7334914 0.84 KLK5 (0.57) BACE1CTSDKLK5
SCHEMBL7269733 0.83 KLK5 (0.55) BACE1CTSDKLK5
SCHEMBL6449655 0.83 CTSD (0.66) BACE1CTSDKLK5
SCHEMBL7270592 0.82 KLK5 (0.63) KLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed