SCHEMBL8540529

SCHEMBL8540529

OC(c1ccccc1)(c1ccccc1)[C@H]1OC(c2ccccc2)O[C@@H]1C(O)(c1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
LMNA P02545 2/20 0.40
HRH1 P35367 1/20 0.40
SCN1A P35498 1/20 0.40
SCN2A Q99250 1/20 0.40
SCN3A Q9NY46 1/20 0.40
CYP2C19 P33261 3/20 0.37
CYP1A2 P05177 2/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
CHRM3 P20309 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.34
ATM Q13315 1/20 0.34
EPHX1 P07099 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8537818 1.00 MAPK1 (0.50) MAPK1CYP3A4CYP2D6MEN1KMT2A
SCHEMBL19784271 0.74 MEN1 (0.39) MAPK1CYP3A4MEN1KMT2ALMNA
SCHEMBL25954641 0.74 MEN1 (0.39) MAPK1CYP3A4MEN1KMT2ALMNA
SCHEMBL125445 0.74 MEN1 (0.39) MAPK1CYP3A4MEN1KMT2ALMNA
SCHEMBL9199389 0.73 MAPK1 (0.53) MAPK1CYP3A4CYP2D6MEN1KMT2A
SCHEMBL20702256 0.73 EPHX1 (0.44) MAPK1CYP3A4CYP2D6LMNACYP2C19
SCHEMBL6495554 0.70 MAPK1 (0.53) MAPK1CYP3A4CYP2D6MEN1KMT2A
SCHEMBL16309629 0.68 CYP3A4 (0.77) MAPK1CYP3A4CYP2D6MEN1KMT2A
SCHEMBL19419092 0.67 MEN1 (0.45) MEN1KMT2ALMNACYP2C19L3MBTL1
SCHEMBL12393860 0.67 SIRT1 (0.49) MAPK1CYP3A4MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0358154-B1 Novel cyclobutane derivative and process for producing same NIPPON KAYAKU KK (JP) 1998-12-02 EP disclosed
US-5250697-A Drugs, perfumes, reagents, intermediates for viraicides NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1993-10-05 US disclosed
EP-0444597-A1 Novel cyclobutane derivative Nippon Kayaku Kabushiki Kaisha (JP) 1991-09-04 EP disclosed