SCHEMBL8540531

SCHEMBL8540531

O=C1CCc2cc(C(O)CN3CCCC(Cc4ccccc4)C3)ccc2N1

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 4/20 0.62
KCNH2 Q12809 2/20 0.51
OGT O15294 2/20 0.49
ALDH1A1 P00352 1/20 0.46
ATM Q13315 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
KDM4E B2RXH2 1/20 0.43
S1PR1 P21453 1/20 0.42
S1PR3 Q99500 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8541679 1.00 GRIN2B (0.62) GRIN2BKCNH2OGTALDH1A1ATM
SCHEMBL8547979 1.00 GRIN2B (0.62) GRIN2BKCNH2OGTALDH1A1ATM
SCHEMBL8547850 1.00 GRIN2B (0.62) GRIN2BKCNH2OGTALDH1A1ATM
Hydrochloric Acid SCHEMBL8548360 0.94 GRIN2B (0.55) GRIN2BKCNH2OGTALDH1A1ATM
Hydrochloric Acid SCHEMBL8548193 0.94 GRIN2B (0.55) GRIN2BKCNH2OGTALDH1A1ATM
SCHEMBL8547674 0.93 GRIN2B (0.55) GRIN2BKCNH2OGTMAOAMAOB
SCHEMBL8872102 0.93 GRIN2B (0.55) GRIN2BKCNH2OGTMAOAMAOB
SCHEMBL8546412 0.88 GRIN2B (0.50) GRIN2BKCNH2OGTMAOAMAOB
SCHEMBL8548698 0.86 GRIN2B (0.47) GRIN2BKCNH2ALDH1A1ATMMEN1
SCHEMBL8547693 0.86 GRIN2B (0.47) GRIN2BKCNH2ALDH1A1ATMMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709384-B1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GMBH (DE) 1998-12-23 EP claimed
US-5698553-A Benzylpiperidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-16 US claimed
EP-0709384-A1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GmbH (DE) 1996-05-01 EP claimed
JP-8225569-A None JP disclosed
EP-0709384-B1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GMBH (DE) 1998-12-23 EP disclosed
US-5698553-A Benzylpiperidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-16 US disclosed
JP-H08225569-A BENZYLPIPERIDINE DERIVATIVE MERCK PATENT GMBH 1996-09-03 JP disclosed
EP-0709384-A1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GmbH (DE) 1996-05-01 EP disclosed