SCHEMBL8540629

SCHEMBL8540629

c1cc2c(c(-c3ncc[nH]3)c1)OCO2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTBK1 Q5TCY1 1/20 0.43
TTBK2 Q6IQ55 1/20 0.43
CSNK1A1 P48729 1/20 0.41
TYRO3 Q06418 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
NISCH Q9Y2I1 3/20 0.40
MTOR P42345 1/20 0.40
ADK P55263 1/20 0.40
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
RIPK3 Q9Y572 1/20 0.38
CHEK1 O14757 1/20 0.38
CHEK2 O96017 1/20 0.38
ADRA1A P35348 2/20 0.37
CASP6 P55212 1/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.35
ADRA2A P08913 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7594061 0.75 ABCG2 (0.55) TTBK1TTBK2RIPK3CHEK1CHEK2
SCHEMBL10657892 0.74 RIPK3 (0.38) TTBK1TTBK2MEN1ALDH1A1KMT2A
SCHEMBL26259965 0.72 NISCH (0.54) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL9287236 0.71 NISCH (0.64) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL4347210 0.70 RIPK3 (0.56) ALDH1A1RIPK3CHEK1CHEK2PKM
SCHEMBL28382846 0.70 CSNK1A1 (0.56) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL2977832 0.70 PDE10A (0.44) CSNK1A1TYRO3DYRK1BMEN1ALDH1A1
SCHEMBL14886257 0.69 NISCH (0.61) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL10780010 0.69 NISCH (0.51) NISCHADRA2AADRA2C
SCHEMBL768730 0.68 NISCH (0.42) CSNK1A1TYRO3DYRK1BNISCHMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed