SCHEMBL8545286

SCHEMBL8545286

O=C1C=C(Cc2ccccc2)C(=O)C(S)=C1Cc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.53
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
TEK Q02763 1/20 0.44
MEN1 O00255 2/20 0.42
NSD2 O96028 2/20 0.42
KMT2A Q03164 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
MAPK1 P28482 1/20 0.40
HIF1A Q16665 1/20 0.40
PARK7 Q99497 1/20 0.40
CALM1 P0DP23 1/20 0.37
XIAP P98170 2/20 0.35
CTRC Q99895 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2515239 0.75 MAOA (0.69) PTPN1MAOAMAOBTEKMEN1
SCHEMBL9588537 0.74 PTPN1 (0.76) PTPN1MAOAMAOBTEKMEN1
SCHEMBL11322423 0.69 PTPN1 (1.00) PTPN1MAOAMAOBTEKMEN1
SCHEMBL28166599 0.67 PTPN1 (0.42) PTPN1MAOAMAOBTEKMEN1
SCHEMBL27623517 0.66 MAOA (0.57) PTPN1MAOAMAOBCYP1A2CYP2C9
SCHEMBL28800705 0.66 CYP2C9 (0.47) PTPN1MAOAMAOBTEKMEN1
SCHEMBL17969811 0.66 PTPN1 (0.62) PTPN1MAOAMAOBTEKMEN1
SCHEMBL16938333 0.65 BACE1 (0.57) PTPN1MAOAMAOBMEN1NSD2
SCHEMBL1872240 0.64 MAOA (1.00) PTPN1MAOAMAOBTEKPARK7
SCHEMBL27936013 0.64 PTPN1 (0.56) PTPN1MAOAMAOBTEKMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827501-A INERT TRIARYLMETHYL FREE RADICAL CONTRAST AGENTS FOR ELECTRON SPIN RESONANCE (ESR) ENHANCED MAGNETIC RESONANCE (EMR) IMAGING NYCOMED IMAGING AS (NO) 1998-10-27 US disclosed
US-5599522-A CONTRAST ENHANCING AGENTS NYCOMED IMAGING AS (NO) 1997-02-04 US disclosed
EP-0515458-B1 TRIARYLMETHYL RADICALS AND THE USE OF INERT CARBON FREE RADICALS IN MRI NYCOMED INNOVATION AB (SE) 1995-08-23 EP disclosed
EP-0515458-A1 TRIARYLMETHYL RADICALS AND THE USE OF INERT CARBON FREE RADICALS IN MRI. HAFSLUND NYCOMED INNOVATION (SE) 1992-12-02 EP disclosed
WO-1991012024-A1 TRIARYLMETHYL RADICALS AND THE USE OF INERT CARBON FREE RADICALS IN MRI HAFSLUND NYCOMED INNOVATION AB (SE) 1991-08-22 WO disclosed