SCHEMBL8545581

SCHEMBL8545581

CC(C)(C)OC(=O)N1CCC(COC(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)(c2ccccc2)CC1

nearest known ligand 0.72

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.72
SLC6A4 P31645 3/20 0.48
CCR5 P51681 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8107943 0.85 TACR1 (0.55) TACR1SLC6A4
SCHEMBL5216125 0.84 TACR1 (1.00) TACR1SLC6A4
SCHEMBL8544652 0.82 TACR1 (0.69) TACR1SLC6A4
SCHEMBL8824347 0.82 TACR1 (0.72) TACR1SLC6A4
SCHEMBL8546545 0.81 TACR1 (0.66) TACR1SLC6A4
SCHEMBL8540809 0.81 TACR1 (0.68) TACR1SLC6A4
SCHEMBL8824359 0.80 TACR1 (0.73) TACR1SLC6A4
SCHEMBL8824352 0.80 TACR1 (0.73) TACR1SLC6A4
SCHEMBL8561630 0.80 TACR1 (0.67) TACR1SLC6A4
SCHEMBL6482875 0.80 TACR1 (0.59) TACR1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739336-B1 GEM-DISUBSTITUTED AZACYCLIC TACHYKININ ANTAGONISTS MERCK SHARP & DOHME (GB) 1998-08-26 EP disclosed