SCHEMBL8561630

SCHEMBL8561630

COC(=O)CC(C)(OCC1(c2ccccc2)CCN(C(=O)OC(C)(C)C)CC1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.67
SLC6A4 P31645 3/20 0.45
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8545581 0.80 TACR1 (0.72) TACR1SLC6A4
SCHEMBL5216125 0.80 TACR1 (1.00) TACR1SLC6A4
SCHEMBL8546545 0.79 TACR1 (0.66) TACR1SLC6A4
SCHEMBL8562729 0.79 TACR1 (0.70) TACR1SLC6A4
SCHEMBL17886658 0.79 TACR1 (0.63) TACR1ALOX15TSHR
SCHEMBL8544652 0.78 TACR1 (0.69) TACR1SLC6A4
SCHEMBL8540809 0.77 TACR1 (0.68) TACR1SLC6A4
SCHEMBL8824359 0.77 TACR1 (0.73) TACR1SLC6A4
SCHEMBL8824352 0.77 TACR1 (0.73) TACR1SLC6A4
SCHEMBL13543974 0.76 TACR1 (0.55) TACR1ALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760018-A Gem-disubstituted azacyclic tachykinin antagonists MERCK SHARP & DOHME LTD. (GB) 1998-06-02 US disclosed
WO-1995019344-A1 GEM-DISUBSTITUTED AZACYCLIC TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1995-07-20 WO disclosed