Dimethylamine

Dimethylamine

SCHEMBL8545876

CCCNC(=O)c1nccc2c(C)c3[nH]c4ccc(OC)cc4c3cc12.CNC

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.55
BCHE P06276 3/20 0.46
KDM4E B2RXH2 5/20 0.45
MAPT P10636 3/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
RAB9A P51151 2/20 0.45
POLB P06746 2/20 0.45
TLR3 O15455 1/20 0.45
NR3C1 P04150 1/20 0.45
PKM P14618 1/20 0.45
RECQL P46063 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HPGD P15428 2/20 0.44
ACHE P22303 1/20 0.44
DYRK1A Q13627 1/20 0.44
ALDH1A1 P00352 3/20 0.43
NPC1 O15118 1/20 0.43
BRAF P15056 2/20 0.42
MTNR1A P48039 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24276997 0.98 KIT (0.57) KITBCHEKDM4EMAPTMEN1
Dimethylamine SCHEMBL8547837 0.93 KIT (0.54) KITBCHEKDM4EMAPTMEN1
SCHEMBL24277000 0.91 KIT (0.54) KITBCHEKDM4EMAPTMEN1
SCHEMBL24277001 0.91 KIT (0.57) KITBCHEKDM4EMAPTMEN1
SCHEMBL24277005 0.90 KIT (0.54) KITBCHEKDM4EMAPTMEN1
SCHEMBL8547834 0.88 KIT (0.56) KITBCHEKDM4EMAPTMEN1
Dimethylamine SCHEMBL8550040 0.88 KIT (0.44) KITKDM4EBRAFNQO2
SCHEMBL9091811 0.86 KIT (0.59) KITBCHEKDM4EMAPTMEN1
SCHEMBL9091784 0.85 KDM4E (0.54) KITBCHEKDM4EMAPTMEN1
SCHEMBL9091805 0.83 KIT (0.53) KITBCHEKDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0591058-B1 Ellipticine derivatives with antitumor activity ADIR (FR) 1998-06-03 EP disclosed
US-5498611-A ANTITUMOR AGENTS ADIR ET COMPAGNIE (FR) 1996-03-12 US disclosed
US-5407940-A Antitumor agents ADIR ET COMPAGNIE (FR) 1995-04-18 US disclosed
EP-0591058-A1 Ellipticine derivatives with antitumor activity ADIR ET COMPAGNIE (FR) 1994-04-06 EP disclosed