SCHEMBL8548568

SCHEMBL8548568

O=c1[nH]c2cc(Cl)c(C(O)CCN3CCC[C@H](Cc4ccccc4)C3)cc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 2/20 0.46
PRMT6 Q96LA8 2/20 0.46
BCHE P06276 1/20 0.43
GRIN1 Q05586 4/20 0.42
GRIN2B Q13224 5/20 0.42
GRIN2D O15399 2/20 0.42
GRIN3B O60391 2/20 0.42
GRIN2A Q12879 2/20 0.42
GRIN2C Q14957 2/20 0.42
GRIN3A Q8TCU5 2/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
HTR2A P28223 2/20 0.39
CCR3 P51677 2/20 0.39
CCR2 P41597 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8544887 1.00 CARM1 (0.46) CARM1PRMT6BCHEGRIN1GRIN2B
SCHEMBL8546790 0.89 GRIN2B (0.54) GRIN1GRIN2BGRIN2DGRIN3BGRIN2A
SCHEMBL8587995 0.89 CARM1 (0.46) CARM1PRMT6BCHEGRIN1GRIN2B
SCHEMBL8543189 0.89 CARM1 (0.46) CARM1PRMT6BCHEGRIN1GRIN2B
SCHEMBL8872814 0.87 MEN1 (0.47) CARM1PRMT6BCHEGRIN1GRIN2B
SCHEMBL8546732 0.87 MEN1 (0.47) CARM1PRMT6BCHEGRIN1GRIN2B
SCHEMBL8548361 0.87 MEN1 (0.47) CARM1PRMT6BCHEGRIN1GRIN2B
SCHEMBL8542181 0.85 GRIN2B (0.52) CARM1PRMT6BCHEGRIN1GRIN2B
SCHEMBL8873050 0.85 GRIN2B (0.52) CARM1PRMT6BCHEGRIN1GRIN2B
SCHEMBL8547812 0.85 GRIN2B (0.52) CARM1PRMT6BCHEGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709384-B1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GMBH (DE) 1998-12-23 EP disclosed
US-5698553-A Benzylpiperidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-16 US disclosed
EP-0709384-A1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GmbH (DE) 1996-05-01 EP disclosed