SCHEMBL8548583

SCHEMBL8548583

Cc1cc(C)c(S(=O)(=O)NC(CNC(=O)C2CC(CCCCN(C)c3ncc[nH]3)ON2)C(=O)O)c(C)c1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 17/20 0.52
ITGA2B P08514 17/20 0.52
ITGAV P06756 17/20 0.52
ITGB1 P05556 2/20 0.44
ITGA5 P08648 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7396351 0.86 ITGB3 (0.70) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7401670 0.85 ITGB3 (0.70) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7407597 0.84 ITGB3 (0.69) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL8548575 0.83 ITGB3 (0.76) ITGB3ITGA2BITGAV
Trifluoroacetic Acid SCHEMBL7403171 0.83 ITGB3 (0.65) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7403223 0.80 ITGB3 (0.69) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7982597 0.80 ITGB3 (0.71) ITGB3ITGA2BITGAV
SCHEMBL7404741 0.79 ITGB3 (0.55) ITGB3ITGA2BITGAV
SCHEMBL7402546 0.79 ITGAV (0.53) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7397410 0.77 ITGB3 (0.53) ITGB3ITGA2BITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828737-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-03-18 EP disclosed