SCHEMBL8548588

SCHEMBL8548588

CCOC(=O)Oc1c(-c2ccc3nsnc3c2)c2cc(N(C(N)=O)c3ccccc3)ccc2n1Cc1ccccc1OC

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 11/20 0.40
EDNRA P25101 2/20 0.38
ABL1 P00519 1/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
RIN1 Q13671 1/20 0.34
PLA2G2A P14555 7/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549342 0.90 EDNRB (0.45) EDNRBEDNRAMAPTMAPK1PLA2G2A
SCHEMBL8549812 0.87 EDNRB (0.41) EDNRBEDNRAPLA2G2A
SCHEMBL8552678 0.87 EDNRB (0.43) EDNRBEDNRAABL1MAPTMAPK1
SCHEMBL8552533 0.87 EDNRB (0.52) EDNRBEDNRAPLA2G2A
SCHEMBL8547912 0.85 EDNRB (0.43) EDNRBEDNRAMAPTPLA2G2A
SCHEMBL8549391 0.84 EDNRB (0.44) EDNRBEDNRAMAPTMAPK1PLA2G2A
SCHEMBL8546593 0.83 EDNRB (0.42) EDNRBEDNRAPLA2G2A
SCHEMBL8549027 0.80 EDNRB (0.49) EDNRBEDNRAMAPTPLA2G2A
SCHEMBL8551802 0.80 EDNRB (0.39) EDNRBEDNRAMAPT
SCHEMBL8553153 0.79 EDNRB (0.43) EDNRBEDNRAMAPTPLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed