SCHEMBL8551802

SCHEMBL8551802

CCOC(=O)Oc1c(-c2ccc3nsnc3c2)c2cc([N+](=O)[O-])ccc2n1Cc1ccccc1OC.COc1ccccc1CCl

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 8/20 0.39
ELANE P08246 2/20 0.37
EDNRA P25101 1/20 0.36
SERPINE1 P05121 1/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPC1 O15118 1/20 0.34
NPBWR1 P48145 1/20 0.34
RAB9A P51151 1/20 0.34
MCHR1 Q99705 1/20 0.34
F2 P00734 1/20 0.34
PLAU P00749 1/20 0.34
CTRB1 P17538 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552639 0.88 EDNRB (0.43) EDNRBELANEEDNRAALDH1A1MAPT
SCHEMBL8552494 0.85 EDNRB (0.49) EDNRBELANEEDNRAF2PLAU
SCHEMBL8551818 0.85 EDNRB (0.41) EDNRBEDNRAALDH1A1MAPT
SCHEMBL8552678 0.85 EDNRB (0.43) EDNRBEDNRAMAPTNPC1RAB9A
SCHEMBL8547749 0.84 EDNRB (0.41) EDNRBEDNRAALDH1A1
SCHEMBL8552487 0.84 EDNRB (0.44) EDNRBEDNRAMAPT
SCHEMBL8552520 0.83 EDNRB (0.46) EDNRBELANEEDNRAF2PLAU
SCHEMBL8546118 0.83 EDNRB (0.42) EDNRBELANEEDNRAMEN1KMT2A
SCHEMBL8548809 0.81 EDNRB (0.54) EDNRBELANEEDNRAF2PLAU
SCHEMBL8548588 0.80 EDNRB (0.40) EDNRBEDNRAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed