SCHEMBL8548591

SCHEMBL8548591

Nc1ccc2occ(C3CCNCC3)c2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.39
HTR6 P50406 2/20 0.36
HTR1A P08908 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
ADRB2 P07550 1/20 0.36
DRD2 P14416 1/20 0.35
SLC6A4 P31645 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
QDPR P09417 1/20 0.35
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
NPC1 O15118 2/20 0.34
MAPT P10636 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29688867 0.82 KCNH2 (0.45) HTR2CHTR6HTR1ASLC6A4NPC1
SCHEMBL29688968 0.82 HTR2C (0.46) HTR2CHTR6HTR1ADRD2SLC6A4
SCHEMBL4491304 0.82 KCNH2 (0.45) HTR2CHTR6HTR1ASLC6A4NPC1
SCHEMBL4503187 0.82 HTR2C (0.46) HTR2CHTR6HTR1ADRD2SLC6A4
Hydrochloric Acid SCHEMBL8916365 0.81 HTR2C (0.47) HTR2CHTR6HTR1ADRD2SLC6A4
Hydrochloric Acid SCHEMBL7694678 0.81 MPO (0.46) HTR2CHTR6HTR1ASLC6A4
SCHEMBL8548177 0.79 HTR1D (0.56) HTR1DHTR1BDRD2SLC6A4CHRNB2
SCHEMBL7967288 0.78 PTPN1 (0.44) HTR2CHTR6DRD2SLC6A4CHRNB2
SCHEMBL13584551 0.78 SLC6A4 (0.55) HTR2CHTR6HTR1AADRB2DRD2
SCHEMBL20809221 0.75 HTR2C (0.49) HTR2CHTR1AADRB2DRD2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed