SCHEMBL8548669

SCHEMBL8548669

COc1ccccc1C1(O)CCC(c2ccccc2)(c2ccccc2)C2CN(C(=O)Cc3ccccc3O)CC21

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.64
FNTA P49354 7/20 0.56
FNTB P49356 7/20 0.56
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
SIGMAR1 Q99720 1/20 0.40
GRIN2B Q13224 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8956927 1.00 TACR1 (0.64) TACR1FNTAFNTBKMT2AMEN1
SCHEMBL8545840 0.93 TACR1 (0.67) TACR1FNTAFNTBKMT2AMEN1
SCHEMBL8956909 0.93 TACR1 (0.67) TACR1FNTAFNTBKMT2AMEN1
SCHEMBL8956845 0.88 TACR1 (0.68) TACR1FNTAFNTBKMT2AMEN1
SCHEMBL8957044 0.88 TACR1 (0.68) TACR1FNTAFNTBKMT2AMEN1
SCHEMBL8957083 0.88 TACR1 (0.68) TACR1FNTAFNTBKMT2AMEN1
SCHEMBL8956789 0.88 TACR1 (0.61) TACR1FNTAFNTBKMT2AMEN1
SCHEMBL8956777 0.88 TACR1 (0.63) TACR1FNTAFNTBKMT2AMEN1
SCHEMBL8956821 0.88 TACR1 (0.61) TACR1FNTAFNTBKMT2AMEN1
SCHEMBL7582580 0.87 TACR1 (0.66) TACR1FNTAFNTBKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635003-B1 PERHYDROISOINDOLE DERIVATIVES AS P SUBSTANCE ANTAGONISTS RHONE POULENC RORER SA (FR) 1998-06-17 EP claimed
US-5484804-A Perhydroisoindole derivatives as antagonists of substance P RHONE-POULENC RORER S.A. (FR) 1996-01-16 US claimed
US-5484804-A Perhydroisoindole derivatives as antagonists of substance P RHONE-POULENC RORER S.A. (FR) 1996-01-16 US disclosed