SCHEMBL8549161

SCHEMBL8549161

O=C1C(=O)c2c3ccccc3c(Cl)c3cccc1c23

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 3/20 0.54
ALDH1A1 P00352 4/20 0.42
CES2 O00748 2/20 0.42
BCHE P06276 2/20 0.42
MCL1 Q07820 1/20 0.42
DNMT1 P26358 3/20 0.42
IDO1 P14902 1/20 0.39
DNMT3L Q9UJW3 1/20 0.39
DNMT3A Q9Y6K1 1/20 0.39
CYP1A2 P05177 3/20 0.39
MAPT P10636 6/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
PABPC1 P11940 4/20 0.39
KDM4E B2RXH2 3/20 0.39
POLB P06746 4/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
LMNA P02545 2/20 0.38
PTPRC P08575 2/20 0.38
S100A4 P26447 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8542998 0.79 TYMS (0.54) CES1ALDH1A1DNMT1IDO1DNMT3L
SCHEMBL587124 0.78 CES1 (0.54) CES1ALDH1A1CES2BCHEMCL1
SCHEMBL3183695 0.78 CES1 (0.54) CES1ALDH1A1CES2BCHEMCL1
SCHEMBL14257731 0.74 CES1 (0.46) CES1ALDH1A1CES2BCHEMCL1
SCHEMBL12179533 0.73 CES1 (0.49) CES1ALDH1A1CES2BCHEMCL1
SCHEMBL8845047 0.71 DNMT1 (0.54) CES1ALDH1A1CES2BCHEMCL1
SCHEMBL12179771 0.70 CES1 (0.50) CES1ALDH1A1CES2BCHEMCL1
SCHEMBL12179578 0.70 CES1 (0.50) CES1ALDH1A1CES2BCHEMCL1
SCHEMBL2156357 0.70 CES1 (1.00) CES1ALDH1A1CES2BCHEMCL1
SCHEMBL579274 0.70 CES1 (1.00) CES1ALDH1A1CES2BCHEMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536208-B1 1,2-DIHYDRO-3H-DIBENZISOQUINOLINE-1,3-DIONE ANTICANCER AGENTS RES CORP TECHNOLOGIES INC (US) 1998-01-21 EP disclosed
US-5635506-A ANTITUMOR AGENTS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1997-06-03 US disclosed
EP-0660824-A1 1,2 DIHYDRO-3-H-DIBENZ(de,h) ISOQUINOLINE 1,3 DIONE AND THEIR USE AS ANTICANCER AGENTS RESEARCH CORPORATION TECHNOLOGIES (US) 1995-07-05 EP disclosed
WO-1994006771-A9 1,2 DIHYDRO-3-H-DIBENZ(de,h) ISOQUINOLINE 1,3 DIONE AND THEIR USE AS ANTICANCER AGENTS 1994-06-09 WO disclosed
WO-1994006771-A1 1,2 DIHYDRO-3-H-DIBENZ(de,h) ISOQUINOLINE 1,3 DIONE AND THEIR USE AS ANTICANCER AGENTS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1994-03-31 WO disclosed
EP-0536208-A4 1,2-DIHYDRO-3H-DIBENZISOQUINOLINE-1,3-DIONE ANTICANCER AGENTS 1993-05-05 EP disclosed
EP-0536208-A1 1,2-DIHYDRO-3H-DIBENZISOQUINOLINE-1,3-DIONE ANTICANCER AGENTS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1993-04-14 EP disclosed
WO-1992000281-A1 1,2-DIHYDRO-3H-DIBENZISOQUINOLINE-1,3-DIONE ANTICANCER AGENTS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1992-01-09 WO disclosed