Oxalic Acid

Oxalic Acid

SCHEMBL8549166

COc1ccc2[nH]cc(CCN)c2c1Cl.O=C(O)C(=O)O

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.56
MTNR1A P48039 2/20 0.45
MTNR1B P49286 2/20 0.45
NQO2 P16083 1/20 0.45
CYP1A2 P05177 3/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTR1A P08908 5/20 0.44
HTR2C P28335 3/20 0.44
HTR7 P34969 3/20 0.44
HTR1D P28221 3/20 0.44
HTR1B P28222 3/20 0.44
TRPM8 Q7Z2W7 2/20 0.44
TSHR P16473 2/20 0.44
HTR6 P50406 2/20 0.44
MAPT P10636 1/20 0.44
NFKB1 P19838 1/20 0.44
HTR4 Q13639 1/20 0.44
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2541508 0.92 HTR2A (0.65) HTR2ACYP1A2HTR1AHTR2CHTR7
Fumaric Acid SCHEMBL8549914 0.92 HTR2A (0.53) HTR2AMTNR1AMTNR1BNQO2CYP1A2
Fumaric Acid SCHEMBL8549920 0.92 HTR2A (0.53) HTR2AMTNR1AMTNR1BNQO2CYP1A2
SCHEMBL8545521 0.80 HTR2A (0.44) HTR2ACYP1A2CYP2C9CYP2C19HTR1A
Fumaric Acid SCHEMBL8549291 0.79 HTR1A (0.47) HTR2AMTNR1AMTNR1BNQO2CYP1A2
Fumaric Acid SCHEMBL8549290 0.79 HTR1A (0.47) HTR2AMTNR1AMTNR1BNQO2CYP1A2
Fumaric Acid SCHEMBL8549603 0.78 HTR1A (0.46) HTR2ACYP1A2CYP2C9CYP2C19HTR1A
Fumaric Acid SCHEMBL8549599 0.78 HTR1A (0.46) HTR2ACYP1A2CYP2C9CYP2C19HTR1A
SCHEMBL8546978 0.78 HTR2A (0.50) HTR2ACYP1A2HTR1AHTR2CHTR7
Fumaric Acid SCHEMBL8543245 0.78 HTR1A (0.59) HTR2AMTNR1AMTNR1BNQO2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0593513-B1 TRYPTAMINE ANALOGUES, THEIR SYNTHESIS AND THEIR USE AS 5-HT1-LIKE RECEPTORS OR 5-HT2 RECEPTOR AGONISTES SMITHKLINE BEECHAM PLC (GB) 1998-10-28 EP disclosed
US-5571833-A TREATMENT OF MIGRAINE, PORTAL HYPERTENSION SMITHKLINE BEECHAM PLC (GB) 1996-11-05 US disclosed
EP-0593513-A1 TRYPTAMINE ANALOGUES, THEIR SYNTHESIS AND THEIR USE AS 5-HT1-LIKE RECEPTORS OR 5-HT2 RECEPTOR AGONISTES SMITHKLINE BEECHAM PLC (GB) 1994-04-27 EP disclosed
WO-1993000333-A1 TRYPTAMINE ANALOGUES, THEIR SYNTHESIS AND THEIR USE AS 5-HT1-LIKE OR 5-HT2 RECEPTOR AGONISTS SMITHKLINE BEECHAM PLC (GB) 1993-01-07 WO disclosed