SCHEMBL8549192

SCHEMBL8549192

CC(C)(C)OC(=O)N1[C@H](C(=O)N2CCCC2)C[C@@H]2CCCC[C@@H]21

nearest known ligand 0.56

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PREP P48147 11/20 0.56
HPGD P15428 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9321884 1.00 PREP (0.56) PREPHPGD
SCHEMBL9321893 1.00 PREP (0.56) PREPHPGD
SCHEMBL9177599 0.99 PREP (0.55) PREPHPGD
SCHEMBL9323315 0.99 PREP (0.55) PREPHPGD
SCHEMBL9323319 0.99 PREP (0.55) PREPHPGD
SCHEMBL9183787 0.97 PREP (0.53) PREPHPGD
SCHEMBL8313638 0.84 PREP (0.42) PREPHPGD
SCHEMBL4840543 0.83 CHRM2 (0.45) PREP
SCHEMBL4795338 0.83 CHRM2 (0.45) PREPHPGD
SCHEMBL1336739 0.83 CHRM2 (0.45) PREP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618193-B1 Nitrogen containing bicyclic derivatives as prolyl-endopeptidase inhibitors ADIR (FR) 1998-10-21 EP disclosed
US-5506237-A PROLYL-ENDOPEPTIDASE INHIBITOR; USEFUL FOR TREATING OR PREVENTING MEMORY LOSS DUE TO AGING, ANXIETY AND DEPRESSION ADIR ET COMPAGNIE (FR) 1996-04-09 US disclosed
US-5384322-A Prolylendopeptidase inhibitors; Alzheimer*s disease; antidepressant and anxiolytic agents ADIR ET COMPAGNIE (FR) 1995-01-24 US disclosed
EP-0618193-A1 Nitrogen containing bicyclic derivatives as prolyl-endopeptidase inhibitors ADIR ET COMPAGNIE (FR) 1994-10-05 EP disclosed