SCHEMBL8549745

SCHEMBL8549745

O=C(O)c1ccc2c(c1)CCOC2CCO[C@H]1CCCCO1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
HTR1D P28221 14/20 0.41
HTR1B P28222 7/20 0.41
DRD2 P14416 5/20 0.41
HTR2A P28223 5/20 0.41
HTR1A P08908 3/20 0.41
DRD4 P21917 2/20 0.41
KDM4C Q9H3R0 1/20 0.39
CREBBP Q92793 2/20 0.38
SLC6A4 P31645 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.36
EP300 Q09472 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8812246 1.00 MEN1 (0.55) MEN1KMT2AHTR1DHTR1BDRD2
SCHEMBL8811219 0.84 MEN1 (0.39) MEN1KMT2AHTR1DHTR1BDRD2
SCHEMBL8551017 0.84 MEN1 (0.39) MEN1KMT2AHTR1DHTR1BDRD2
SCHEMBL6812077 0.79 HTR1D (0.43) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL5097946 0.79 HTR1D (0.43) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL8550172 0.79 HTR1D (0.46) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL2981986 0.72 MEN1 (0.88) MEN1KMT2AKDM4CCREBBPL3MBTL1
SCHEMBL12193490 0.71 KMT2A (0.67) MEN1KMT2AKDM4CRAB9A
SCHEMBL7385130 0.71 MEN1 (0.51) MEN1KMT2ACREBBPEP300
SCHEMBL224651 0.71 MEN1 (1.00) MEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed
WO-1997002259-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1997-01-23 WO disclosed