SCHEMBL8551017

SCHEMBL8551017

CN(OCc1ccccc1)C(=O)c1ccc2c(c1)CCOC2CCO[C@H]1CCCCO1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HTR1D P28221 8/20 0.38
HTR1B P28222 3/20 0.38
DRD2 P14416 5/20 0.36
HTR2A P28223 5/20 0.36
HTR1A P08908 3/20 0.36
DRD4 P21917 2/20 0.36
THRB P10828 1/20 0.35
KDM4C Q9H3R0 2/20 0.35
ALDH1A1 P00352 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPT P10636 2/20 0.35
EP300 Q09472 1/20 0.35
CREBBP Q92793 1/20 0.35
OXTR P30559 1/20 0.35
AVPR1A P37288 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8811219 1.00 MEN1 (0.39) MEN1KMT2AHTR1DHTR1BDRD2
SCHEMBL8551173 0.84 HTR1D (0.41) MEN1KMT2AHTR1DHTR1BDRD2
SCHEMBL8549745 0.84 MEN1 (0.55) MEN1KMT2AHTR1DHTR1BDRD2
SCHEMBL8812246 0.84 MEN1 (0.55) MEN1KMT2AHTR1DHTR1BDRD2
SCHEMBL8551680 0.74 HTR1D (0.66) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL6811827 0.69 HTR1D (0.42) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL6811442 0.68 HTR1D (0.42) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL6811669 0.68 HTR1D (0.42) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL6808728 0.67 HTR1D (0.45) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL5097946 0.67 HTR1D (0.43) HTR1DHTR1BDRD2HTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed
WO-1997002259-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1997-01-23 WO disclosed