SCHEMBL8549747

SCHEMBL8549747

COc1ccc(N2CCN(CCC3OCCc4cc(C(=O)NCc5ccccc5)ccc43)CC2)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 8/20 0.78
DRD2 P14416 7/20 0.78
HTR2A P28223 7/20 0.78
DRD4 P21917 6/20 0.78
HTR1A P08908 5/20 0.78
HTR1B P28222 1/20 0.78
SLC6A4 P31645 1/20 0.54
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
PPARG P37231 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
NR2E3 Q9Y5X4 1/20 0.49
NCOR2 Q9Y618 1/20 0.49
ADRA2A P08913 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
DRD1 P21728 1/20 0.49
ADRA1D P25100 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methane SCHEMBL8596364 0.99 HTR1D (0.77) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8550481 0.96 HTR1D (0.81) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8550881 0.90 DRD2 (0.75) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8550141 0.90 HTR1D (0.84) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8552917 0.89 HTR1D (0.76) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8550001 0.89 HTR1D (0.80) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8810266 0.88 HTR1D (0.81) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8621436 0.88 HTR1D (0.81) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL5595821 0.88 HTR1D (1.00) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL7401976 0.88 HTR1D (1.00) HTR1DDRD2HTR2ADRD4HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed
WO-1997002259-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1997-01-23 WO claimed
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed