SCHEMBL8549877

SCHEMBL8549877

O=Cc1cc2c(N3CCN(CCc4ccccc4)CC3)cccc2s1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 10/20 0.54
DRD2 P14416 9/20 0.54
HTR2A P28223 8/20 0.54
MEN1 O00255 1/20 0.51
ALDH1A1 P00352 1/20 0.51
KMT2A Q03164 1/20 0.51
CYP2C9 P11712 1/20 0.51
SIGMAR1 Q99720 1/20 0.48
ADRA1D P25100 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48
SLC6A4 P31645 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9213148 0.85 HTR1A (0.52) HTR1ADRD2HTR2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL6017140 0.84 CYP2C9 (0.47) HTR1ADRD2HTR2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL8550533 0.84 CYP2C9 (0.47) HTR1ADRD2HTR2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL6017220 0.83 HTR1A (0.49) HTR1ADRD2HTR2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL8550861 0.83 HTR1A (0.49) HTR1ADRD2HTR2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL6017185 0.83 CYP2C9 (0.46) HTR1ADRD2HTR2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL8546875 0.83 CYP2C9 (0.46) HTR1ADRD2HTR2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL8550912 0.82 HTR1A (0.48) HTR1ADRD2HTR2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL8550906 0.82 HTR1A (0.48) HTR1ADRD2HTR2AMEN1ALDH1A1
SCHEMBL8544808 0.81 MEN1 (0.51) HTR1ADRD2HTR2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660832-B1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMA INC (US) 1998-01-14 EP disclosed
US-5436246-A Compounds for treatment of anxiety, depression, migraine, stroke, angina and hypertension MERRELL DOW PHARMACEUTICALS INC. 1995-07-25 US disclosed
EP-0660832-A1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMACEUTICALS INC. (US) 1995-07-05 EP disclosed
WO-1994006789-A1 SEROTONIN RECEPTOR AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-31 WO disclosed