SCHEMBL8550171

SCHEMBL8550171

NC(=O)c1ccc2c(c1)CCOC2CCN1CCC(c2ccccc2)CC1

nearest known ligand 0.76

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 20/20 0.76
HTR1B P28222 11/20 0.76
DRD2 P14416 3/20 0.61
HTR2A P28223 3/20 0.61
HTR1A P08908 3/20 0.61
DRD4 P21917 1/20 0.61
SLC6A4 P31645 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8811237 0.88 HTR1D (0.67) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL6812051 0.86 HTR1D (1.00) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL8551188 0.86 HTR1D (0.78) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL27563581 0.84 HTR1D (0.78) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL5090663 0.84 HTR1D (0.78) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL8554794 0.83 HTR1D (0.53) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL7408003 0.82 DRD2 (0.61) HTR1DHTR1BDRD2HTR2AHTR1A
Hydrochloric Acid SCHEMBL7406756 0.81 DRD2 (0.60) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL6811594 0.81 HTR1D (0.82) HTR1DHTR1BDRD2HTR1ASLC6A4
SCHEMBL6812692 0.81 HTR1D (0.82) HTR1DHTR1BDRD2HTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed