SCHEMBL8550179

SCHEMBL8550179

N#Cc1ccc(Oc2cccc(Oc3ccc(C#N)cc3Cl)c2)c(Cl)c1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.60
CYP19A1 P11511 1/20 0.53
KCNH2 Q12809 3/20 0.49
SLC6A4 P31645 2/20 0.49
HTR2A P28223 2/20 0.49
MRGPRX4 Q96LA9 4/20 0.48
SLC6A3 Q01959 1/20 0.47
EGFR P00533 1/20 0.46
ERBB2 P04626 1/20 0.46
ERBB3 P21860 1/20 0.46
ERBB4 Q15303 1/20 0.46
FFAR1 O14842 1/20 0.46
EPAS1 Q99814 3/20 0.46
ICMT O60725 2/20 0.45
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10088434 0.90 AR (0.65) ARCYP19A1KCNH2SLC6A4HTR2A
SCHEMBL4171609 0.89 AR (0.70) ARCYP19A1KCNH2SLC6A4HTR2A
SCHEMBL11088375 0.89 AR (0.54) ARCYP19A1KCNH2SLC6A4HTR2A
SCHEMBL4168829 0.85 MRGPRX4 (0.50) ARCYP19A1KCNH2SLC6A4HTR2A
SCHEMBL2747584 0.83 EGFR (0.50) ARCYP19A1KCNH2SLC6A4HTR2A
SCHEMBL3258951 0.83 EGFR (0.47) ARCYP19A1KCNH2SLC6A4HTR2A
SCHEMBL920869 0.81 AR (0.54) ARCYP19A1KCNH2SLC6A4HTR2A
SCHEMBL13875516 0.81 AR (0.62) ARKCNH2SLC6A4HTR2ASLC6A3
SCHEMBL10852120 0.80 AR (0.54) ARKCNH2SLC6A4HTR2AMRGPRX4
SCHEMBL14334473 0.80 AR (0.54) ARCYP19A1KCNH2SLC6A4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696585-B1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMA CO LTD (JP) 1998-12-16 EP disclosed
US-5643931-A ANTIDIABETIC AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1997-07-01 US disclosed
EP-0696585-A1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-02-14 EP disclosed