SCHEMBL8550465

SCHEMBL8550465

COc1ccc(C2CCN(CCC3OCCc4cc(Br)ccc43)CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 10/20 0.55
DRD2 P14416 8/20 0.55
HTR2A P28223 6/20 0.55
HTR1A P08908 4/20 0.55
DRD4 P21917 3/20 0.55
HTR1B P28222 4/20 0.53
KCNH2 Q12809 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8809830 1.00 HTR1D (0.55) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL8554794 0.86 HTR1D (0.53) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL8591943 0.86 DRD2 (0.74) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL7403729 0.86 DRD2 (0.74) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL8590932 0.86 DRD2 (0.74) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL7401836 0.85 DRD2 (0.74) HTR1DDRD2HTR2AHTR1ADRD4
Hydrochloric Acid SCHEMBL7403803 0.85 DRD2 (0.73) HTR1DDRD2HTR2AHTR1ADRD4
Hydrochloric Acid SCHEMBL8185555 0.85 DRD2 (0.72) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL8548563 0.82 HTR1D (0.78) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL8550170 0.82 HTR1D (0.78) HTR1DDRD2HTR2AHTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed
WO-1997002259-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1997-01-23 WO disclosed