SCHEMBL8550705

SCHEMBL8550705

C[Si](C)(C)CCOCn1nccc1C(=O)c1ccccc1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.38
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
HSD17B10 Q99714 8/20 0.36
ALDH1A1 P00352 8/20 0.36
CFTR P13569 1/20 0.35
KDM4E B2RXH2 3/20 0.34
POLB P06746 1/20 0.34
TP53 P04637 3/20 0.34
ALOX15 P16050 1/20 0.34
HPGD P15428 4/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
MAPK1 P28482 2/20 0.34
ESRRA P11474 3/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
RAB9A P51151 2/20 0.33
GLA P06280 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550681 0.82 NPC1 (0.39) NPC1GAAMAPTALDH1A1KDM4E
SCHEMBL30415291 0.79 NPC1 (0.43) NPC1MAPTALDH1A1HPGDSMN1; SMN2
SCHEMBL8543053 0.79 NPC1 (0.36) NPC1GAAMAPTHSD17B10ALDH1A1
SCHEMBL1288508 0.78 NPC1 (0.36) NPC1MAPTALDH1A1HPGDSMN1; SMN2
SCHEMBL30785205 0.78 KLKB1 (0.38) NPC1MAPTALDH1A1HPGDSMN1; SMN2
SCHEMBL8544222 0.77 NPC1 (0.36) NPC1GAAMAPTHSD17B10ALDH1A1
SCHEMBL8543719 0.75 ESRRA (0.38) NPC1GAAMAPTHSD17B10ALDH1A1
SCHEMBL30414625 0.74 F2RL1 (0.38) NPC1GAAALDH1A1KDM4EPOLB
SCHEMBL19332634 0.72 KDM4E (0.42) NPC1ALDH1A1KDM4EPOLB
SCHEMBL29110304 0.70 F2RL1 (0.33) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0715624-B1 PROCESS FOR THE PREPARATION OF BENZODIAZEPINE COMPOUNDS USEFUL AS ANTAGONISTS OF CCK OR OF GASTRINE YAMANOUCHI PHARMA CO LTD (JP) 1998-04-08 EP disclosed
US-5728829-A MULTISTAGE REACTION OF N-PROTECTED BENZOTRIAZOLYL GLYCINE DERIVATIVE WITH AMINOKETONE, THEN REACTION WITH AMMONIA AND ACID CATALYZED CYCLIZATION FERRING-RESEARCH LIMITED (GB) 1998-03-17 US disclosed
WO-1995006040-A1 BENZODIAZEPINE COMPOUNDS USEFUL AS ANTAGONISTS OF CCK OR OF GASTRINE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-02 WO disclosed