SCHEMBL8550681

SCHEMBL8550681

C[Si](C)(C)CCOCn1nccc1C(=O)c1ccccc1[N+](=O)[O-]

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
CTSD P07339 1/20 0.38
HTT P42858 4/20 0.37
HPGD P15428 2/20 0.37
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
GAA P10253 1/20 0.36
NCOA1 Q15788 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NCOA3 Q9Y6Q9 1/20 0.36
LMNA P02545 1/20 0.36
MEN1 O00255 1/20 0.36
ESRRA P11474 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8544025 0.79 MET (0.38) NPC1RAB9ACTSDHTTHPGD
SCHEMBL8544357 0.77 ESRRA (0.39) NPC1RAB9ACTSDHTTHPGD
SCHEMBL1288508 0.74 NPC1 (0.36) NPC1RAB9AHTTHPGDKMT2A
SCHEMBL30785205 0.74 KLKB1 (0.38) NPC1RAB9AHPGDKMT2AALDH1A1
SCHEMBL19332428 0.73 F2RL1 (0.33) NPC1
SCHEMBL30415291 0.73 NPC1 (0.43) NPC1RAB9AHTTHPGDKMT2A
SCHEMBL9685754 0.73 KMT2A (0.42) HTTHPGDKMT2AALDH1A1MAPT
SCHEMBL4718604 0.71 TDP1 (0.37) NPC1RAB9AHTTKMT2AALDH1A1
SCHEMBL29258063 0.71 ALDH1A1 (0.37) NPC1RAB9AHTTALDH1A1GAA
SCHEMBL9038725 0.71 ALDH1A1 (0.39) NPC1RAB9ACTSDHTTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0715624-B1 PROCESS FOR THE PREPARATION OF BENZODIAZEPINE COMPOUNDS USEFUL AS ANTAGONISTS OF CCK OR OF GASTRINE YAMANOUCHI PHARMA CO LTD (JP) 1998-04-08 EP disclosed
US-5728829-A MULTISTAGE REACTION OF N-PROTECTED BENZOTRIAZOLYL GLYCINE DERIVATIVE WITH AMINOKETONE, THEN REACTION WITH AMMONIA AND ACID CATALYZED CYCLIZATION FERRING-RESEARCH LIMITED (GB) 1998-03-17 US disclosed
WO-1995006040-A1 BENZODIAZEPINE COMPOUNDS USEFUL AS ANTAGONISTS OF CCK OR OF GASTRINE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-02 WO disclosed