SCHEMBL8550792

SCHEMBL8550792

N#Cc1cccc2c(-c3ccccc3)nnc(Cl)c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
NPSR1 Q6W5P4 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
CYP1A2 P05177 3/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 3/20 0.39
KDM4E B2RXH2 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MAPT P10636 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
PDE5A O76074 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
PDE1A P54750 1/20 0.39
PDE1B Q01064 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE1C Q14123 1/20 0.39
PDE3A Q14432 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551333 0.87 ALDH1A1 (0.41) ALDH1A1NPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL31488270 0.82 DYRK1A (0.40) ALDH1A1NPSR1TDP1CYP1A2CYP2C9
SCHEMBL8548327 0.79 ALDH1A1 (0.43) ALDH1A1NPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL8550823 0.78 ALDH1A1 (0.42) ALDH1A1NPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL8552241 0.76 ALDH1A1 (0.41) ALDH1A1NPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL8549262 0.76 ALDH1A1 (0.41) ALDH1A1NPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL8552220 0.75 PLG (0.42) ALDH1A1KDM4ESMN1; SMN2MAPTMAP2K1
SCHEMBL8552217 0.73 KDM4E (0.37) ALDH1A1NPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL8548189 0.73 NPSR1 (0.41) ALDH1A1NPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL8546259 0.73 NR1H2 (0.41) ALDH1A1NPSR1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed