SCHEMBL8551173

SCHEMBL8551173

CN(OCc1ccccc1)C(=O)c1ccc2c(c1)CCO[C@H]2CCO

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 8/20 0.41
HTR1B P28222 3/20 0.41
THRB P10828 1/20 0.41
DRD2 P14416 5/20 0.41
HTR2A P28223 5/20 0.41
HTR1A P08908 3/20 0.41
DRD4 P21917 2/20 0.41
ALDH1A1 P00352 4/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
MAPT P10636 4/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
BLM P54132 1/20 0.38
KDM4E B2RXH2 1/20 0.38
TP53 P04637 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8811219 0.84 MEN1 (0.39) HTR1DHTR1BTHRBDRD2HTR2A
SCHEMBL8551017 0.84 MEN1 (0.39) HTR1DHTR1BTHRBDRD2HTR2A
SCHEMBL6808728 0.83 HTR1D (0.45) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL20906508 0.82 HTR1D (0.43) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL8551680 0.81 HTR1D (0.66) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL8550172 0.78 HTR1D (0.46) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL20921215 0.77 HTR1D (0.41) HTR1DHTR1BTHRBDRD2HTR2A
SCHEMBL20921241 0.77 HTR1D (0.41) HTR1DHTR1BTHRBDRD2HTR2A
SCHEMBL6812048 0.75 HTR1D (0.56) HTR1DHTR1BDRD2HTR2AHTR1A
SCHEMBL5093578 0.75 HTR1D (0.56) HTR1DHTR1BDRD2HTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed
WO-1997002259-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1997-01-23 WO disclosed