SCHEMBL8551193

SCHEMBL8551193

COc1cc2nccc(Oc3ccc(N(C(N)=S)c4ccccc4F)cc3)c2cc1OC

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 9/20 0.55
KDR P35968 6/20 0.55
PDGFRB P09619 1/20 0.54
FGFR2 P21802 4/20 0.53
KIT P10721 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552680 0.90 PDGFRA (0.54) PDGFRAKDRPDGFRBFGFR2KIT
SCHEMBL8556665 0.90 PDGFRA (0.59) PDGFRAKDRPDGFRBFGFR2KIT
SCHEMBL8552480 0.88 PDGFRA (0.67) PDGFRAKDRPDGFRBFGFR2KIT
SCHEMBL31105478 0.84 KDR (0.55) PDGFRAKDRKIT
SCHEMBL8554464 0.82 PDGFRA (0.56) PDGFRAKDRPDGFRBFGFR2
SCHEMBL8554120 0.82 PDGFRA (0.58) PDGFRAKDRPDGFRBFGFR2KIT
SCHEMBL8554994 0.80 PDGFRA (0.57) PDGFRAKDRPDGFRBFGFR2KIT
SCHEMBL8552659 0.80 PDGFRA (0.67) PDGFRAKDRPDGFRBFGFR2KIT
SCHEMBL8551093 0.79 AXL (0.56) PDGFRAKDRPDGFRBFGFR2KIT
SCHEMBL8555319 0.79 PDGFRA (0.63) PDGFRAKDRPDGFRBFGFR2KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP disclosed