SCHEMBL8552680

SCHEMBL8552680

COc1cc2nccc(Oc3ccc(N(C(N)=S)c4ccccc4C)cc3)c2cc1OC

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 7/20 0.54
PDGFRB P09619 1/20 0.54
KDR P35968 2/20 0.53
FGFR2 P21802 4/20 0.53
KIT P10721 3/20 0.51
AXL P30530 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551193 0.90 PDGFRA (0.55) PDGFRAPDGFRBKDRFGFR2KIT
SCHEMBL5825546 0.87 PDGFRA (0.59) PDGFRAPDGFRBKDRFGFR2KIT
SCHEMBL8554464 0.84 PDGFRA (0.56) PDGFRAPDGFRBKDRFGFR2
SCHEMBL8552480 0.84 PDGFRA (0.67) PDGFRAPDGFRBKDRFGFR2KIT
SCHEMBL8554120 0.82 PDGFRA (0.58) PDGFRAPDGFRBKDRFGFR2KIT
SCHEMBL8556665 0.80 PDGFRA (0.59) PDGFRAPDGFRBKDRFGFR2KIT
SCHEMBL5825989 0.79 PDGFRA (0.61) PDGFRAPDGFRBKDRFGFR2KIT
SCHEMBL8555506 0.78 KDR (0.57) PDGFRAPDGFRBKDRFGFR2AXL
SCHEMBL8552489 0.78 PDGFRA (0.65) PDGFRAPDGFRBKDRFGFR2KIT
SCHEMBL5826134 0.78 PDGFRA (0.66) PDGFRAPDGFRBKDRFGFR2KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP disclosed