SCHEMBL8551196

SCHEMBL8551196

COc1ccc(-c2c(OC(=O)O)n(Cc3ccc4nsnc4c3)c3cccc(OC)c23)cc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 6/20 0.52
EDNRA P25101 2/20 0.47
PLA2G2A P14555 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
MEN1 O00255 2/20 0.37
MAPT P10636 2/20 0.37
KMT2A Q03164 2/20 0.37
HTT P42858 2/20 0.37
GAA P10253 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
CNR2 P34972 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CCR2 P41597 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553011 0.93 EDNRB (0.51) EDNRBEDNRAPLA2G2AKDM4EALDH1A1
SCHEMBL8549015 0.92 EDNRB (0.50) EDNRBEDNRASMN1; SMN2MAPTHTT
SCHEMBL8553494 0.91 EDNRB (0.52) EDNRBEDNRASMN1; SMN2NPC1RAB9A
SCHEMBL8547582 0.90 EDNRB (0.52) EDNRBEDNRASMN1; SMN2NPC1RAB9A
SCHEMBL8551194 0.88 EDNRB (0.64) EDNRBEDNRAPLA2G2A
SCHEMBL8550887 0.88 EDNRB (0.58) EDNRBEDNRASMN1; SMN2NPC1RAB9A
SCHEMBL8552686 0.86 EDNRB (0.53) EDNRBEDNRASMN1; SMN2NPC1RAB9A
SCHEMBL8547527 0.85 EDNRB (0.48) EDNRBEDNRASMN1; SMN2NPC1RAB9A
SCHEMBL8549175 0.85 EDNRB (0.59) EDNRBEDNRAGAA
SCHEMBL8550230 0.84 EDNRB (0.66) EDNRBEDNRAPLA2G2ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed