SCHEMBL8551276

SCHEMBL8551276

COc1ccc(-c2c(C(=O)O)n(Cc3ccc4nsnc4c3)c3cc(OCc4ccccc4)ccc23)cc1F

nearest known ligand 0.61

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 16/20 0.61
EDNRA P25101 13/20 0.58
TP53 P04637 1/20 0.42
S1PR3 Q99500 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551759 0.93 EDNRB (0.62) EDNRBEDNRATP53
SCHEMBL8552951 0.91 EDNRB (0.66) EDNRBEDNRA
SCHEMBL8553793 0.90 EDNRB (0.70) EDNRBEDNRATP53
SCHEMBL8551281 0.90 EDNRB (0.49) EDNRBEDNRAS1PR3
SCHEMBL8551612 0.89 EDNRB (0.58) EDNRBEDNRATP53
SCHEMBL8552334 0.87 EDNRB (0.73) EDNRBEDNRA
SCHEMBL8551430 0.87 EDNRB (0.80) EDNRBEDNRA
SCHEMBL8549140 0.87 EDNRB (0.48) EDNRBEDNRAS1PR3
SCHEMBL8547973 0.86 EDNRB (0.75) EDNRBEDNRA
SCHEMBL8547214 0.86 EDNRB (0.56) EDNRBEDNRATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed