SCHEMBL8551297

SCHEMBL8551297

Cc1ccc(NC(=O)CCCCCCBr)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.73
HDAC1 Q13547 3/20 0.73
HDAC2 Q92769 3/20 0.73
HDAC10 Q969S8 3/20 0.73
HDAC11 Q96DB2 2/20 0.73
HDAC8 Q9BY41 2/20 0.73
HDAC6 Q9UBN7 2/20 0.73
NCOR2 Q9Y618 1/20 0.73
HDAC4 P56524 1/20 0.71
HDAC7 Q8WUI4 1/20 0.71
HDAC9 Q9UKV0 1/20 0.71
HDAC5 Q9UQL6 1/20 0.71
POLB P06746 3/20 0.60
ALDH1A1 P00352 3/20 0.59
LMNA P02545 2/20 0.59
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
NSD2 O96028 1/20 0.54
ABL1 P00519 1/20 0.54
MAPK1 P28482 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15883219 0.98 HDAC3 (0.73) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL23540107 0.93 HDAC3 (0.70) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL517697 0.89 HDAC3 (0.86) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL29111436 0.86 HDAC1 (0.56) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL19962693 0.86 POLB (0.68) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL17252159 0.85 HDAC3 (0.76) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL2531377 0.85 HDAC3 (0.76) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL2319941 0.85 HDAC3 (0.76) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL22479429 0.85 MEN1 (0.61) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL13524769 0.85 HDAC1 (1.00) HDAC3HDAC1HDAC2HDAC10HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660832-B1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMA INC (US) 1998-01-14 EP disclosed
US-5436246-A Compounds for treatment of anxiety, depression, migraine, stroke, angina and hypertension MERRELL DOW PHARMACEUTICALS INC. 1995-07-25 US disclosed
EP-0660832-A1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMACEUTICALS INC. (US) 1995-07-05 EP disclosed
WO-1994006789-A1 SEROTONIN RECEPTOR AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-31 WO disclosed