SCHEMBL8551475

SCHEMBL8551475

COc1ccc(-c2c(C(=O)O)n(Cc3ccc4nsnc4c3)c3cc(OCc4ccccc4)c(OC)cc23)c(OC)c1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 16/20 0.58
EDNRA P25101 12/20 0.58
TP53 P04637 2/20 0.41
PLK1 P53350 1/20 0.41
POLB P06746 1/20 0.41
CSF1R P07333 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552564 0.93 EDNRB (0.66) EDNRBEDNRATP53POLB
SCHEMBL8547214 0.91 EDNRB (0.56) EDNRBEDNRATP53POLB
SCHEMBL8551023 0.91 EDNRB (0.67) EDNRBEDNRATP53PLK1CSF1R
SCHEMBL8549315 0.89 EDNRB (0.64) EDNRBEDNRATP53POLB
SCHEMBL8551476 0.89 EDNRB (0.48) EDNRBEDNRAPLK1POLBCSF1R
SCHEMBL8552951 0.85 EDNRB (0.66) EDNRBEDNRACSF1R
SCHEMBL8550894 0.85 EDNRB (0.59) EDNRBEDNRATP53
SCHEMBL8548858 0.85 EDNRB (0.45) EDNRBEDNRAPLK1POLBCSF1R
SCHEMBL8550885 0.83 EDNRB (0.74) EDNRBEDNRATP53
SCHEMBL8548412 0.83 EDNRB (0.62) EDNRBEDNRATP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed