SCHEMBL8551548

SCHEMBL8551548

COC(=O)Nc1ccc2c(c1)c(-c1ccc(C=O)cc1)c(OC(=O)O)n2Cc1ccc2nsnc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 5/20 0.46
EDNRA P25101 2/20 0.42
KDM4E B2RXH2 3/20 0.35
SERPINE1 P05121 3/20 0.34
NPC1 O15118 5/20 0.34
SMN1; SMN2 Q16637 5/20 0.34
RAB9A P51151 4/20 0.34
MAPT P10636 4/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
GAA P10253 1/20 0.34
TSHR P16473 2/20 0.33
ATM Q13315 1/20 0.33
HSD17B10 Q99714 1/20 0.33
LMNA P02545 3/20 0.33
HTT P42858 2/20 0.33
TP53 P04637 2/20 0.32
POLB P06746 2/20 0.32
SCD O00767 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549437 0.91 EDNRB (0.48) EDNRBEDNRAKDM4ESERPINE1NPC1
SCHEMBL8548371 0.91 EDNRB (0.44) EDNRBEDNRAKDM4ESERPINE1NPC1
SCHEMBL8551480 0.91 EDNRB (0.57) EDNRBEDNRAKDM4ENPC1SMN1; SMN2
SCHEMBL8546737 0.88 EDNRB (0.49) EDNRBEDNRAKDM4ENPC1SMN1; SMN2
SCHEMBL8551727 0.87 EDNRB (0.47) EDNRBEDNRASERPINE1MAPT
SCHEMBL8550751 0.85 EDNRB (0.46) EDNRBEDNRAKDM4ESERPINE1SMN1; SMN2
SCHEMBL8551102 0.85 EDNRB (0.45) EDNRBEDNRAKDM4ESERPINE1MEN1
SCHEMBL8548022 0.85 EDNRB (0.44) EDNRBEDNRAKDM4ENPC1SMN1; SMN2
SCHEMBL8548304 0.83 EDNRB (0.44) EDNRBEDNRAKDM4ENPC1SMN1; SMN2
SCHEMBL8550822 0.83 EDNRB (0.66) EDNRBEDNRAKDM4EGAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed