SCHEMBL8551728

SCHEMBL8551728

Cc1nc(CCCOc2c(C)cc(-c3nnn(C)n3)cc2C)cs1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
PKM P14618 1/20 0.34
FABP6 P51161 1/20 0.33
SMN1; SMN2 Q16637 4/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
EPHX2 P34913 1/20 0.33
MAPT P10636 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8603712 0.81 NR1I2 (0.37) NR1I2CYP3A4CYP2D6SMN1; SMN2NPC1
SCHEMBL8824410 0.80 NR1I2 (0.35) NR1I2CYP3A4CYP2D6SMN1; SMN2NPC1
SCHEMBL8824405 0.80 NPC1 (0.34) NR1I2CYP3A4CYP2D6SMN1; SMN2NPC1
SCHEMBL9089930 0.79 NR1I2 (0.35) NR1I2CYP3A4CYP2D6SMN1; SMN2NPC1
SCHEMBL8553801 0.79 NR1I2 (0.35) NR1I2CYP3A4CYP2D6PKMSMN1; SMN2
SCHEMBL8556856 0.78 NR1I2 (0.33) NR1I2CYP3A4CYP2D6SMN1; SMN2NPC1
SCHEMBL8992121 0.78 BRD4 (0.37) NR1I2CYP3A4CYP2D6SMN1; SMN2NPC1
SCHEMBL8552613 0.77 NR1I2 (0.47) NR1I2CYP3A4CYP2D6FABP6SMN1; SMN2
SCHEMBL8553780 0.77 NPC1 (0.36) NR1I2CYP3A4CYP2D6SMN1; SMN2NPC1
SCHEMBL8605399 0.76 NR1I2 (0.36) NR1I2CYP3A4CYP2D6SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5846986-A Therapeutic phenoxyalkylazoles and phenoxyalkylazines SANOFI (FR) 1998-12-08 US disclosed
US-5721261-A TREATING PICORNAVIRUS INFECTIONS SANOFI PHARMACEUTICALS, INC. (US) 1998-02-24 US disclosed