SCHEMBL8552140

SCHEMBL8552140

OC(CCc1cccnc1)COc1ccc(-c2ccc(F)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 1/20 0.43
ADRB1 P08588 2/20 0.43
ADRB3 P13945 2/20 0.43
ADRB2 P07550 1/20 0.43
ELOVL1 Q9BW60 1/20 0.43
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
MMP12 P39900 1/20 0.41
CYP3A4 P08684 3/20 0.39
SIGMAR1 Q99720 1/20 0.39
NPC1 O15118 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP19A1 P11511 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
CACNA1G O43497 2/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8476865 1.00 MEN1 (0.45) MEN1KMT2AALDH1A1ADRB1ADRB3
SCHEMBL8479732 0.90 MEN1 (0.52) MEN1KMT2AALDH1A1ADRB1ADRB3
SCHEMBL8477371 0.90 CYP19A1 (0.50) MEN1KMT2AALDH1A1ADRB1ADRB3
SCHEMBL8109540 0.90 MEN1 (0.52) MEN1KMT2AALDH1A1ADRB1ADRB3
SCHEMBL8481421 0.90 MEN1 (0.52) MEN1KMT2AALDH1A1ADRB1ADRB3
SCHEMBL8483060 0.90 MEN1 (0.42) MEN1KMT2AALDH1A1ADRB1ADRB3
SCHEMBL8118428 0.90 MEN1 (0.42) MEN1KMT2AALDH1A1ADRB1ADRB3
SCHEMBL8118260 0.90 MEN1 (0.42) MEN1KMT2AALDH1A1ADRB1ADRB3
SCHEMBL7829887 0.88 MEN1 (0.45) MEN1KMT2AALDH1A1ADRB1ADRB3
SCHEMBL8482114 0.88 NPC1 (0.48) MEN1KMT2AALDH1A1ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed