SCHEMBL8552163

SCHEMBL8552163

CCSc1cc(C(F)(F)F)c(-n2ccnc2)cc1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
CYP1A2 P05177 3/20 0.45
CYP3A4 P08684 3/20 0.45
CYP2D6 P10635 3/20 0.45
CYP2C19 P33261 3/20 0.45
LMNA P02545 2/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C9 P11712 1/20 0.45
MAPK1 P28482 1/20 0.45
PMP22 Q01453 1/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
DDR1 Q08345 1/20 0.33
CYP19A1 P11511 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
IDO1 P14902 2/20 0.33
ADH5 P11766 2/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3495779 0.70 CYP1A2 (0.51) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL12017706 0.67 CYP1A2 (0.62) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL3496197 0.66 GRIK1 (0.53) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL994454 0.64 CYP1A2 (0.62) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL15011268 0.64 ALDH1A1 (0.50) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL27294485 0.64 CYP1A2 (0.62) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL12015798 0.64 ALDH1A1 (0.57) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL8139118 0.64 GRIA1 (0.67) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL251863 0.64 CYP1A2 (0.57) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL29595684 0.63 CYP3A4 (1.00) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877191-A ANTIINFLAMMATORY AGENT; ANALGESICS; ANTIHISTAMINES; EMESIS MERCK & CO., INC. (US) 1999-03-02 US disclosed
WO-1998017660-A1 PHENYL SPIROETHERCYCLOALKYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1998-04-30 WO disclosed