SCHEMBL8552519

SCHEMBL8552519

Cc1nc(-c2ccc(Cl)cc2)c(-c2ccc(S(N)(=O)=O)cc2)o1

nearest known ligand 0.76

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.76
PTGS1 P23219 12/20 0.76
MAOA P21397 1/20 0.55
MAOB P27338 1/20 0.55
CA12 O43570 2/20 0.50
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA9 Q16790 2/20 0.50
CA3 P07451 1/20 0.50
CA4 P22748 1/20 0.50
CA6 P23280 1/20 0.50
CA5A P35218 1/20 0.50
CA7 P43166 1/20 0.50
CA13 Q8N1Q1 1/20 0.50
CA14 Q9ULX7 1/20 0.50
CA5B Q9Y2D0 1/20 0.50
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7504621 1.00 PTGS2 (0.76) PTGS2PTGS1MAOAMAOBCA12
SCHEMBL7505993 0.93 PTGS2 (0.86) PTGS2PTGS1CA12CA1CA2
SCHEMBL213986 0.87 PTGS2 (0.78) PTGS2PTGS1MAOAMAOBCA12
SCHEMBL8551037 0.87 PTGS2 (0.78) PTGS2PTGS1MAOAMAOBCA12
SCHEMBL7505580 0.86 PTGS2 (1.00) PTGS2PTGS1MAOAMAOBKMT2A
SCHEMBL7799127 0.86 PTGS2 (0.76) PTGS2PTGS1CA12CA1CA2
SCHEMBL8140711 0.86 PTGS2 (0.76) PTGS2PTGS1CA12CA1CA2
SCHEMBL8552366 0.86 PTGS2 (0.76) PTGS2PTGS1CA12CA1CA2
SCHEMBL7500813 0.86 PTGS2 (1.00) PTGS2PTGS1MAOAMAOBKMT2A
SCHEMBL31194859 0.85 MAPK13 (0.57) PTGS2PTGS1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825989-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-03-04 EP claimed
WO-1996036617-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-11-21 WO claimed
EP-0825989-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-03-04 EP disclosed
WO-1996036617-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-11-21 WO disclosed