SCHEMBL8552742

SCHEMBL8552742

CCOC(=O)Oc1c(-c2ccc(C=O)cc2)c2cc([N+](=O)[O-])ccc2n1Cc1ccc2nsnc2c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 3/20 0.43
EDNRA P25101 2/20 0.39
AR P10275 1/20 0.36
PLA2G2A P14555 1/20 0.36
ELANE P08246 1/20 0.36
RAD52 P43351 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
POLB P06746 1/20 0.35
TXNRD1 Q16881 1/20 0.35
TXNRD3 Q86VQ6 1/20 0.35
TXNRD2 Q9NNW7 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548809 0.90 EDNRB (0.54) EDNRBEDNRAPLA2G2AELANE
SCHEMBL8552520 0.88 EDNRB (0.46) EDNRBEDNRAPLA2G2AELANE
SCHEMBL8548805 0.88 EDNRB (0.45) EDNRBEDNRAPLA2G2ASMN1; SMN2
SCHEMBL8552494 0.86 EDNRB (0.49) EDNRBEDNRAELANE
SCHEMBL8548022 0.86 EDNRB (0.44) EDNRBEDNRAELANEMEN1KMT2A
SCHEMBL8546805 0.85 EDNRB (0.61) EDNRBEDNRAPLA2G2A
SCHEMBL8548371 0.84 EDNRB (0.44) EDNRBEDNRAMEN1KMT2ARAB9A
SCHEMBL8546118 0.84 EDNRB (0.42) EDNRBEDNRAPLA2G2AELANEMEN1
SCHEMBL8548911 0.82 EDNRB (0.46) EDNRBEDNRAPLA2G2AELANESMN1; SMN2
SCHEMBL8548322 0.81 EDNRB (0.42) EDNRBEDNRAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed