SCHEMBL8552845

SCHEMBL8552845

Cc1ccc(C(=O)OC2CCN(Cc3ccccc3Br)CC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 2/20 0.57
SCN2A Q99250 2/20 0.57
SCN3A Q9NY46 2/20 0.57
ALDH1A1 P00352 6/20 0.50
KDM4E B2RXH2 3/20 0.50
CARM1 Q86X55 1/20 0.50
PRMT6 Q96LA8 1/20 0.50
LMNA P02545 1/20 0.48
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
MAPT P10636 1/20 0.47
ATM Q13315 1/20 0.46
TSHR P16473 1/20 0.46
RECQL P46063 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
SIGMAR1 Q99720 1/20 0.43
CYP2A13 Q16696 1/20 0.43
FAAH O00519 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8551109 0.99 SCN1A (0.56) SCN1ASCN2ASCN3AALDH1A1KDM4E
SCHEMBL8550475 0.90 ALDH1A1 (0.59) SCN1ASCN2ASCN3AALDH1A1KDM4E
Hydrochloric Acid SCHEMBL8554390 0.89 MEN1 (0.58) SCN1ASCN2ASCN3AALDH1A1KDM4E
SCHEMBL8551519 0.86 SCN1A (0.57) SCN1ASCN2ASCN3AALDH1A1KDM4E
SCHEMBL8553710 0.86 SCN1A (0.57) SCN1ASCN2ASCN3AALDH1A1KDM4E
SCHEMBL8553741 0.86 SCN1A (0.57) SCN1ASCN2ASCN3AALDH1A1KDM4E
Hydrochloric Acid SCHEMBL8551979 0.85 SCN1A (0.56) SCN1ASCN2ASCN3AALDH1A1KDM4E
Hydrochloric Acid SCHEMBL8550203 0.85 SCN1A (0.56) SCN1ASCN2ASCN3AALDH1A1CARM1
Hydrochloric Acid SCHEMBL8554793 0.85 SCN1A (0.56) SCN1ASCN2ASCN3AALDH1A1KDM4E
SCHEMBL8550662 0.83 SCN1A (0.63) SCN1ASCN2ASCN3AALDH1A1CARM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed