SCHEMBL8553551

SCHEMBL8553551

CN(CCN1CCN(c2ccc(C(N)=O)cc2)CC1)C(=O)c1ccc2c(c1)CCOC2

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.48
HTR1D P28221 7/20 0.47
DRD2 P14416 5/20 0.45
HTR2A P28223 5/20 0.45
HTR1A P08908 3/20 0.45
SLC6A4 P31645 1/20 0.40
HRH3 Q9Y5N1 2/20 0.39
HTR1B P28222 1/20 0.38
CHEK1 O14757 1/20 0.38
ADRA2A P08913 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
ADRA1D P25100 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
CHRNA7 P36544 1/20 0.37
CHRNA10 Q9GZZ6 1/20 0.37
CHRNA9 Q9UGM1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551575 0.92 DRD4 (0.48) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8550687 0.92 DRD4 (0.48) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8549471 0.92 DRD4 (0.48) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8550252 0.91 DRD4 (0.59) DRD4DRD2HTR2AHTR1AHRH3
SCHEMBL8550036 0.91 DRD4 (0.47) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8549100 0.91 DRD4 (0.47) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8549609 0.90 DRD4 (0.58) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8551436 0.89 DRD4 (0.48) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8551554 0.89 DRD4 (0.46) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8550849 0.89 DRD4 (0.46) DRD4HTR1DDRD2HTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed