SCHEMBL8550849

SCHEMBL8550849

CN(CCN1CCN(c2ccc(C(=O)C(F)(F)F)cc2)CC1)C(=O)c1ccc2c(c1)CCOC2

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 4/20 0.46
MLYCD O95822 2/20 0.38
HTR1D P28221 7/20 0.38
DRD2 P14416 5/20 0.38
HTR2A P28223 5/20 0.38
HTR1A P08908 4/20 0.38
HRH3 Q9Y5N1 2/20 0.37
HTR1B P28222 1/20 0.36
TACR1 P25103 1/20 0.35
TACR3 P29371 1/20 0.35
SLC6A4 P31645 1/20 0.35
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549843 0.91 DRD4 (0.46) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8551575 0.89 DRD4 (0.48) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8549471 0.89 DRD4 (0.48) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8553551 0.89 DRD4 (0.48) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8550687 0.89 DRD4 (0.48) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8550263 0.89 DRD4 (0.48) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8550252 0.88 DRD4 (0.59) DRD4DRD2HTR2AHTR1AHRH3
SCHEMBL8550036 0.87 DRD4 (0.47) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8549100 0.87 DRD4 (0.47) DRD4HTR1DDRD2HTR2AHTR1A
SCHEMBL8549547 0.87 DRD4 (0.46) DRD4HTR1DDRD2HTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed