SCHEMBL8553580

SCHEMBL8553580

C[C@@H](N(CCOCc1ccccc1)C(=O)c1ccc(OCC(F)(F)C(F)F)cc1)[C@](O)(Cn1cncn1)c1ccc(Cl)cc1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.35
CYP2C9 P11712 6/20 0.35
CYP2C19 P33261 6/20 0.35
CYP1A2 P05177 3/20 0.35
CYP2D6 P10635 3/20 0.35
KCNH2 Q12809 2/20 0.35
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
TP53 P04637 2/20 0.33
PTGS2 P35354 1/20 0.32
LMNA P02545 2/20 0.32
MAPT P10636 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553576 1.00 CYP3A4 (0.35) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8553545 0.89 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9172133 0.89 CYP3A4 (0.36) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8555073 0.89 CYP3A4 (0.39) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8554388 0.87 CYP3A4 (0.39) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8554382 0.87 CYP3A4 (0.39) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8829076 0.83 CYP3A4 (0.48) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8829205 0.80 CYP3A4 (0.46) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8556774 0.77 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8556778 0.77 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0617031-B1 Orally active azole derivates URIACH & CIA SA J (ES) 1998-09-16 EP disclosed
US-5646294-A FUNGICIDES J. URIACH & CIA. S.A. (ES) 1997-07-08 US disclosed
US-5478826-A Fungicides for human, animal and plants J. URIACH & CIA. S.A. (ES) 1995-12-26 US disclosed
EP-0617031-A1 Orally active azole derivates J. URIACH & CIA. S.A. (ES) 1994-09-28 EP disclosed