SCHEMBL8553615

SCHEMBL8553615

O=c1[nH]nc(-c2cccs2)c2sccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 7/20 0.60
ADORA2A P29274 6/20 0.60
HSD17B10 Q99714 2/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
ALDH1A1 P00352 1/20 0.43
ALPL P05186 1/20 0.43
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
GLA P06280 1/20 0.42
CASP1 P29466 1/20 0.42
RAB9A P51151 1/20 0.42
CASP7 P55210 1/20 0.42
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
ATM Q13315 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PKM P14618 1/20 0.39
TYMP P19971 1/20 0.39
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13721415 0.81 ATM (0.59) ADORA2AHSD17B10KDM4EHPGDALDH1A1
SCHEMBL1786973 0.79 NPSR1 (0.62) ADORA1ADORA2AHSD17B10KDM4EHPGD
SCHEMBL14911562 0.78 ADORA1 (0.64) ADORA1ADORA2AHSD17B10KDM4EALDH1A1
SCHEMBL23461929 0.73 ADORA2A (0.53) ADORA1ADORA2AHSD17B10KDM4EALDH1A1
SCHEMBL14633614 0.73 ALDH1A1 (0.43) ADORA1ADORA2AHSD17B10KDM4EHPGD
SCHEMBL24793414 0.73 ADORA2A (0.53) ADORA1ADORA2AHSD17B10KDM4EALDH1A1
SCHEMBL20229834 0.71 ADORA2A (0.55) ADORA1ADORA2AKDM4ENPC1LMNA
SCHEMBL580124 0.71 NPSR1 (0.59) ADORA1ADORA2AKDM4EHPGDALDH1A1
SCHEMBL14611730 0.71 HSD17B10 (0.51) ADORA2AHSD17B10KDM4EHPGDALDH1A1
SCHEMBL4839374 0.71 ENPP1 (0.49) HPGDALDH1A1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0534443-B1 3,6-Disubstituted pyridazine derivatives MITSUBISHI CHEM CORP (JP) 1998-12-30 EP disclosed
US-5462941-A 1-(cyclohexylalkylamino)-4-(phenyl, thienyl, or furyl) phthalazines; anti-platelet agglutination agents for treatment or prevention of cerebro- or cardiovascular disorders MITSUBISHI CHEMICAL CORPORATION (JP) 1995-10-31 US disclosed
EP-0534443-A1 3,6-Disubstituted pyridazine derivatives Mitsubishi Chemical Corporation (JP) 1993-03-31 EP disclosed