SCHEMBL8554230

SCHEMBL8554230

C#CCNC(=O)c1ccc2c(c1)CCOC2CCN1CCN(c2ccc(OC)cc2)CC1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 10/20 0.80
DRD2 P14416 8/20 0.80
HTR2A P28223 6/20 0.80
DRD4 P21917 6/20 0.80
HTR1A P08908 5/20 0.80
HTR1B P28222 3/20 0.80
SLC6A4 P31645 2/20 0.55
ALDH1A1 P00352 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
DRD3 P35462 1/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA4 P22748 1/20 0.47
CA6 P23280 1/20 0.47
CA5A P35218 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550141 0.91 HTR1D (0.84) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8810266 0.89 HTR1D (0.81) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8550481 0.89 HTR1D (0.81) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8621436 0.89 HTR1D (0.81) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL7401976 0.89 HTR1D (1.00) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL5595821 0.89 HTR1D (1.00) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL30628146 0.89 HTR1D (1.00) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8549606 0.89 HTR1D (1.00) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8550530 0.88 HTR1D (0.79) HTR1DDRD2HTR2ADRD4HTR1A
SCHEMBL8812651 0.88 DRD2 (0.79) HTR1DDRD2HTR2ADRD4HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed
WO-1997002259-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1997-01-23 WO claimed
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed